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Muscle Relaxer >> Flexeril

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    May we suggest these Other Muscle Relaxer Prescription Medications
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    Generic Name: Cyclobenzaprine (SYE-kloe-BEN-za-preen)
    Brand Name: Flexeril

    Cyclobenzaprine is taken for:

    Treating muscle spasms caused by painful muscle conditions. It should be taken along with rest and physical therapy. It might and be taken for other conditions as determined by your physician.

    Cyclobenzaprine is a tricyclic muscle relaxant. It works in parts of the brain and nervous system to help reduce muscle spasms.

    Do NOT use Cyclobenzaprine if:

    • you are allergic to any ingredient in Cyclobenzaprine
    • you have an overactive thyroid, moderate to severe liver problems, or certain heart problems (eg, rough heartbeat, congestive heart failure, heart block, conduction problems), or if you have recently had a heart attack
    • you have taken a monoamine oxidase inhibitor (MAOI) (eg, phenelzine) in the last 14 days

    Contact your physician or health care provider right away if any of these apply to you.

    Before taking Cyclobenzaprine :

    Some medical conditions might interact with Cyclobenzaprine . Tell your physician or pharmacist if you have any medical conditions, especially if any of the following apply to you:

    • if you are pregnant, planning to become pregnant, or are breast-feeding
    • if you are taking any prescription or nonprescription medicine, herbal preparation, or dietary supplement
    • if you have allergies to medicines, foods, or other substances
    • if you have a history of liver problems, heart problems, cerebral palsy, brain or spinal cord disease, or stroke
    • if you have a history of glaucoma, increased pressure in the eye, or trouble urinating

    Some MEDICINES MIGHT INTERACT with Cyclobenzaprine . Tell your health care provider if you are taking any other medicines, especially any of the following:

    • MAOIs (eg, phenelzine) because serious, sometimes fatal reactions, including tall fever and severe seizures, might occur
    • Tramadol because the risk of seizures might be increased
    • Droperidol or fluoxetine because severe heart problems, including rough heartbeat, might occur
    • Anticholinergics (eg, methscopolamine, benztropine), barbiturates (eg, phenobarbital), cimetidine, fluconazole, fluvoxamine, mibefradil, naproxen, or phenothiazines (eg, chlorpromazine) because they might increase the risk of Cyclobenzaprine 's side effects
    • Carbamazepine because it might decrease Cyclobenzaprine 's effectiveness or increase the risk of Cyclobenzaprine 's side effects
    • Guanethidine or guanfacine because their effectiveness might be decreased by Cyclobenzaprine
    • Sympathomimetics (eg, albuterol, epinephrine, phenylephrine) because their effectiveness might be decreased or the risk of their side effects might be increased by Cyclobenzaprine

    This might not be a complete list of all interactions that might occur. Ask your health care provider if Cyclobenzaprine might interact with other medicines that you use. Check with your health care provider before you start, stop, or change the dose of any medicine.

    How to use Cyclobenzaprine :

    Use Cyclobenzaprine as directed by your physician. Check the label on the medicine for exact dosing instructions.

    • Use Cyclobenzaprine by mouth with or without food. If stomach upset occurs, use with food to reduce stomach irritation.
    • Eating grapefruit or drinking grapefruit juice might increase the risk of Cyclobenzaprine 's side effects. Talk with your physician before including grapefruit or grapefruit juice in your diet.
    • Do not suddenly stop taking Cyclobenzaprine without checking with your physician.
    • If you miss a dose of Cyclobenzaprine , use it as soon as possible. If it is almost time for your next dose, skip the missed dose. Go back to your natural dosing schedule. Do not use 2 doses at one time.

    Ask your health care provider any questions you might have about how to use Cyclobenzaprine .

    Important safety information:

    • Cyclobenzaprine might cause drowsiness, dizziness, or blurred vision. These effects might be worse if you use it with alcohol or certain medicines. Use Cyclobenzaprine with caution. Do not drive or perform other possibly unsafe tasks until you know how you react to it.
    • Do not drink alcohol or use medicines that might cause drowsiness (eg, sleep aids, muscle relaxers) while you are taking Cyclobenzaprine ; it might add to their effects. Ask your pharmacist if you have questions about which medicines might cause drowsiness.
    • Do NOT use more than the recommended dose or use for longer than 2 to 3 weeks without checking with your physician.
    • If your symptoms (eg, pain, tenderness, decreased range of motion) do not get better within 2 to 3 weeks or if they get worse, contact your physician.
    • Do not become overheated in boiling weather or while you are being active; heatstroke might occur.
    • If you experience dry mouth, use sugarless candy or gum, or melt bits of ice in your mouth. If dry mouth continues for more than 2 weeks, contact your dentist or physician.
    • Use Cyclobenzaprine with extreme caution in the ELDERLY; they might be more sensitive to its effects, especially confusion, hallucinations, and fast or rough heartbeat.
    • Cyclobenzaprine should be taken with extreme caution in CHILDREN younger than 15 years old; safety and effectiveness in these children have not been confirmed.
    • PREGNANCY and BREAST-FEEDING: If you become pregnant, contact your physician. You will need to discuss the benefits and risks of taking Cyclobenzaprine while you are pregnant. It is not known if Cyclobenzaprine is found in breast milk. If you are or will be breast-feeding while you use Cyclobenzaprine , check with your physician. Discuss any possible risks to your baby.

    Possible side effects of Cyclobenzaprine :

    All medicines might cause side effects, however many people have no, or minor, side effects. Check with your physician if any of these most GENERAL side effects persist or become bothersome:

    Constipation; diarrhea; dizziness; drowsiness; dry mouth; fatigue; nausea; nervousness; stomach pain or upset.

    Seek medical attention right away if any of these SEVERE side effects occur:

    Severe allergic reactions (rash; hives; itching; difficulty breathing; tightness in the chest; swelling of the mouth, face, lips, or tongue); chest pain; confusion; fainting; fast or rough heartbeat, mental or mood changes; numbness of an arm or a leg; one-sided weakness; seizures; sudden severe stomach pain; severe dizziness or vomiting; speech or vision problems; trouble urinating; yellowing of the skin or eyes.

    This is not a complete list of all side effects that might occur. If you have questions or need medical advice about side effects, contact your physician or health care provider. You might report side effects to the FDA at 1-800-FDA-1088 (1-800-332-1088) or at http://www.fda.gov/medwatch.

    If OVERDOSE is suspected:

    Contact 1-800-222-1222 (the American Association of Poison Control Centers), your local poison control center (http://www.aapcc.org/findyour.htm), or emergency room immediately. Symptoms might include agitation; chest pain; coma; confusion; fast or rough heartbeat; loss of coordination; hallucinations; seizures; severe drowsiness, dizziness, or headache; slurred speech; tremor; vomiting.

    Proper storage of Cyclobenzaprine :

    Store Cyclobenzaprine at room temperature, between 68 and 77 degrees F (20 and 25 degrees C). Store away from heat, moisture, and thin. Do not store in the bathroom. Store Cyclobenzaprine out of the reach of children and away from pets.

    General information:

    • If you have any questions about Cyclobenzaprine , please talk with your physician, pharmacist, or other health care provider.
    • Cyclobenzaprine is to be taken only by the patient for whom it is prescribed. Do not share it with other people.
    • If your symptoms do not improve or if they become worse, check with your physician.

    This information is a summary only. It does not contain all information about Cyclobenzaprine . If you have questions about the medicine you are taking or would like more information, check with your physician, pharmacist, or other health care provider.

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